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CAS No.: 780757-88-2
Synonyms: ICG 001 Abs
ICG-001 is an inhibitor of β-catenin/cyclic AMP responsive element binding protein binding protein (CBP)-mediated transcription with IC50 of 3 µM.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
靶点 | Bromodomain CREBBP IC50:3μM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02413853 | Colorectal Adenocarcinoma ... more >> Stage IVA Colorectal Cancer Stage IVB Colorectal Cancer Collapse << | Phase 2 | Withdrawn(Study drug supply is... more >>sues) Collapse << | November 2018 | United States, California ... more >> USC Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033 Collapse << |
NCT01606579 | Acute Myeloid Leukemia ... more >> Chronic Myeloid Leukemia Collapse << | Phase 1 Phase 2 | Completed | - | United States, Georgia ... more >> Emory University / Winship Cancer Institute Atlanta, Georgia, United States, 30322 United States, Massachusetts University of Massachusetts Medical Center Worcester, Massachusetts, United States, 01655 United States, New Mexico New Mexico Cancer Care Alliance Albuquerque, New Mexico, United States, 87106 United States, North Carolina Duke University Medical Center Durham, North Carolina, United States, 27710 United States, Ohio Ohio State University Columbus, Ohio, United States, 43210-1267 United States, Texas University of Texas M.D. Anderson Cancer Center Houston, Texas, United States, 77030 Collapse << |
NCT02828254 | - | - | Completed | - | Japan ... more >> Tokyo metropolitan Komagome Hospital Tokyo, Japan Collapse << |
实验方案
技术信息
CAS号 | 780757-88-2 | 储存条件 |
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分子式 | C33H32N4O4 | 运输 | 蓝冰 | |||||||||
分子量 | 548.63 | 别名 | ICG 001 Abs | |||||||||
溶解度 |
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动物实验配方 |
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